Abstract
Easily accessible arylglycine derivatives were cyclized to azetidines by using commercially available (2-bromoethyl)sulfonium triflate in a simple and mild procedure. The high-yielding reaction has a relatively broad scope and was extended to the synthesis of an oxetane.
| Original language | English |
|---|---|
| Pages (from-to) | 1584-1590 |
| Number of pages | 7 |
| Journal | Synthesis (Germany) |
| Volume | 44 |
| Issue number | 10 |
| DOIs | |
| Publication status | Published - May 2012 |
Research Groups and Themes
- Organic & Biological
Keywords
- annulations
- cyclizations
- heterocycles
- sulfur
- ylides
- VINYL SULFONIUM SALTS
- ASYMMETRIC-SYNTHESIS
- DRUG DISCOVERY
- AZETIDINE-2-CARBOXYLIC ACID
- CYCLOPROPANATION REACTIONS
- CONVENIENT METHOD
- CHIRAL CATALYSTS
- TANDEM REACTIONS
- AMINO-ALCOHOLS
- DERIVATIVES
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Dive into the research topics of 'An Efficient Synthesis of Azetidines with (2-Bromoethyl)sulfonium Triflate'. Together they form a unique fingerprint.Projects
- 2 Finished
-
GENERAL AND CONVERGENT STRATEGY FOR ASYMMETRIC SYNTHESIS
Aggarwal, V. K. (Principal Investigator)
1/10/07 → 1/04/13
Project: Research
-
NEW ASSYMETRIC REACTIONS AND THEIR APPLICATION IN TOTAL SYNTHESIS
Aggarwal, V. K. (Principal Investigator)
1/10/05 → 1/10/10
Project: Research
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